Citri•Rx Direct Release Acetyl-Glutathione (100mg)
$94.50 — or subscribe to save 15%
100 mg sublingual format • 120 count
Direct-release troches in a grape flavor. Read the product instructions and ingredients when choosing your supplement format.
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Formerly known as Ovation Acetyl-Glutathione
Healthy Living Protocols:
Using Glutathione : Boost Immunity and Fight Mold Exposure
User Instructions:
We call it a “Troche”
You’ll call it “Incredible”
This innovative “troche” bypasses the bioavailability* problems of oral delivery by going directly to the bloodstream.
This industry-first means lower doses and lower prices for the highest-quality available glutathione supplement, Citri•Rx Sublingual Acetyl-Glutathione.
Glutathione… Simply Delivered.
Sublingual delivery of medicines isn’t rocket science — in fact, it dates back to 1000 BC as an effective way of bypassing the gut. Compound pharmacists have used this delivery method long before the mass production of pharmaceuticals. Today, CitriSafe’s own compounding pharmacist, Walter Hayhurst — a pioneer in sublingual delivery — improves his breakthrough Citri•Rx Acetyl-Glutathione with the simplicity and effectiveness of a sublingual troche. It’s Glutathione. Simply delivered.
Grape Goodness
In a word, our sublingual troche tastes pretty good. When you use a sublingual you place it under your tongue until it dissolves — so you can understand why having a good tasting troche is a big deal. When formulating Citri•Rx Sublingual Acetyl-Glutathione, our pharmacist Walter Hayhurst, took extra care to create a formulation that pleases the palate.
“Simply the best way to take glutathione”
Citri•Rx
Sublingual Acetyl-Glutathione
100 mg | 120 ct

Sublingual administration
Dissolve a Sublingual Acetyl-Glutathione troche underneath the tongue.

Buccal administration
Dissolve a Sublingual Acetyl-Glutathione troche between the gums and cheek.

Sublingual administration
Pour the Glutathione underneath the tongue.

Buccal administration
Pour the Glutathione between the gums and cheek.
Suggested Use: As a dietary supplement, dissolve one troche under your tongue twice daily or as directed by your healthcare professional.
Physician-Grade Quality at Store-Bought Prices
Glutathione Product Comparison Chart
Citri•Rx Compared to:
Other Over-the-Counter Glutathione
1st Generation
L-Glutathione
- Large dosage recommendations 1-3g/day.
- Poor to no bioavailability.
- Eliminated by gut enzymatic processes and water solubility.
- Abundant in food; however, difficult to raise blood levels.
2nd Generation
Liposomal Glutathione, N-Acetyl Cisteine
- Lipids (fat) provide protective layers to guard GHS from digestive processes.
- Enzymatic processes and water solutbility diminish efficacy.
- Large dosing recommendation to allow for diminished active ingredient.
- Wide variation amongst brands.
- Putrid smell due to sulfur.
3rd Generation
Citri•Rx Acetyl-Glutathion
- Over 10 years of product availability.
- Tens of thousands of patients.
- Pharmaceutical grade ingredients (98%+ pure).
- Proprietary nanotech microcluster encapsulation delivers full dose.
- Lower dosing requirements due to improved delivery (100-300mg).
CitriSafe Advantage
A Master Antioxidant Delivered by a Master Laboratory
Enhanced Delivery
using Micro-Cluster Nanotechnology
CitriSafe uses proprietary micro-cluster nanotechnology to employ its glutathione.
Naturally Sourced
from Saccharomyces Cerevisiae
Our Glutathione is naturally sourced from saccharomyces cerevisiae (yeast), not chemically synthesized.
Better Blood Absorption
with Acetylated-Glutathione
Supplementation of Glutathione is challenging due to its poor absorption and water degradation. Acetylated-Glutathione has a more stable molecule improving delivery.
Health Conditions Associated with Low Glutathione
Neuro & Brain
- Alzheimer’s Disease
- Parkinson’s Disease
- Huntington’s Disease
- ALS / Lou Gehrig’s Disease
- Migraines
- Multiple Sclerosis (MS)
- Autism
- ADHD/ADD
- Bipolar Disorder
- Depression
Immune & Cancer
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HIV & AIDS
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Cancer (Breast, Lung, Cervical, Colon, Ovarian, Leukemia)
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Lupus
-
Viral Infections
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Asthma
-
Acne
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Lyme Disease
-
Allergies
-
Gingivitis
-
Rheumatoid Arthritis
Cardiovascular
-
Atherosclerosis
-
Angina
-
Erectile Dysfunction
-
Hypertension
-
Stroke
Thyroid & Pancreas
-
Diabetes
-
Pancreatitis
-
Hyperthyroidism
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Hypothyroidism
Other
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Inflammatory Skin Conditions
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Accelerated Aging
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Arthritis
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Chronic Fatigue
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Chronic Obstructive Pulmonary Disease (COPD)
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Gout
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Hepatitis of Any Kind
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Cystic Fibrosis
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Infertility
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Eyesight Issues
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Gastric Ulcers
FAQs
What makes this different from regular glutathione supplements?
It's a sublingual troche that dissolves under your tongue and absorbs directly into your bloodstream, bypassing the digestive breakdown that destroys most oral glutathione. The acetylated form is more stable than standard L-glutathione, and you only need 100mg twice daily versus the 1-3 grams typical oral supplements require. Developed by compounding pharmacist Walter Hayhurst using nanotech microcluster encapsulation.
Why is this recommended for mold exposure recovery?
Mold exposure depletes your body's glutathione while increasing oxidative stress, and that cycle is hard to break when gut function is already compromised. Sublingual delivery sidesteps the digestive issues common in mold-sensitive individuals. Glutathione directly binds mycotoxins and mold-related free radicals so your body can eliminate them through normal metabolic pathways.
How do I take this?
Dissolve one troche under your tongue and let it sit for two to three minutes. Don't chew or swallow it early. You can also place it between the gums and cheek. Take on an empty stomach and avoid eating, drinking, or brushing your teeth for 15 minutes before and after. Suggested use is one troche twice daily.
Can I adjust the dosage?
The standard recommendation is one troche twice daily for 200mg total. The product supports a range of 100-300mg depending on need, and some practitioners go up to three troches daily for acute situations like severe mold exposure. Work with your healthcare provider on any changes, especially if you're on medications or managing a chronic condition.
Why acetylated glutathione instead of the regular form?
The acetyl group shields the molecule from breaking down during absorption. Standard L-glutathione is vulnerable to oxidation and hydrolysis, which is why oral supplements need such large doses. Once inside your cells, enzymes remove the acetyl group and convert it back to active reduced glutathione. Better stability, better cellular uptake, lower dosing requirements.
What clinical evidence supports this product?
A PMC study found that 150mg of sublingual glutathione produced plasma levels equivalent to 450mg taken orally, with improved GSH/GSSG ratios. The formulation has over 10 years of clinical use. It's manufactured to pharmaceutical-grade standards at 98%+ purity, with third-party testing for potency, composition, and contaminants.
Are there any side effects or drug interactions?
Side effects are minimal. Some people notice mild nausea on a completely empty stomach or slight throat irritation. Glutathione may reduce the effectiveness of certain chemotherapy drugs, so cancer patients should check with their oncologist. Those taking acetaminophen should maintain normal dosing intervals. The product is sourced from yeast, so consult your provider if you have yeast sensitivities.
How does this compare to liposomal glutathione?
Liposomal forms still pass through the digestive tract even with lipid protection. Sublingual delivery skips that entirely for more consistent absorption. Liposomal products often need refrigeration and have shorter shelf lives due to lipid oxidation. These troches stay stable at room temperature for three years. The product page's clinical evidence section notes similar or better bioavailability with sublingual delivery.
How does this compare to NAC supplements?
NAC gives your body cysteine, a building block it uses to make glutathione. That works if your production capacity is intact, but it slows down with age, illness, and toxic burden. This product delivers finished glutathione molecules directly, skipping the synthesis step. Both have therapeutic value and can be used together under practitioner guidance.
How should I store these, and how long do they last?
Room temperature in the original sealed container, away from direct sunlight and humidity. No refrigeration needed. Shelf life is three years when stored properly. The acetylated form and microcluster encapsulation keep the troches stable without the cold storage that some competing glutathione products require.
Many scientific studies have shown and supported the understanding that glutathione has an important role to play in the treatment and prevention of hundreds of diseases. Clinical tests show that raised glutathione levels may address major health issues such as: heart disease, cancer, stroke, diabetes, high cholesterol, asthma, cigarette smoking, hepatitis, AIDS, etc. Glutathione provides the body with tools to fight off these threats naturally. Healthy people also benefit from elevated glutathione levels through an enhanced ability to fight off toxins, infectious disease, pre-cancerous cells and the aging process. Physically active people and world-class athletes are discovering that well-maintained glutathione levels give them the edge over their competitors, providing greater strength and endurance, decreased recovery time from injury, less muscle pain and fatigue, and muscle-promoting activity.
Other Ingredients: Magnesium ascorbate, microcrystalline cellulose, enhanced silica, potassium carbonate, magnesium sulfate, citric acid & fatty acids.
TESTIMONIAL: I want to thank you for introducing me to acetyl glutathione. I have been using it for about four months and have seen numerous remarkable changes to my body and mental processes. I began using it to improve my mold symptoms, which are now essentially gone, but the positive side-effects are truly amazing. Among the changes I've witnessed are the noticeable increase in my muscle mass and hand strength, while my body fat has visibly reduced. My skin and deeper tissue are healing substantially faster than before, and my nails and hair are growing like they did decades ago. In fact, I am beginning to grow new hair after being bald for the past 30 years. I am surprised how important one substance can be to so many aspects of the human body. I can't wait to see how I will be doing after using this item for a year or more. Again, thank you. Best regards, Dr. Dick
TESTIMONIAL: Acetyl-Glutathione is a wonderful treatment for RA. I took Acetyl-Glutathione 100 mg capsules for several years when prescribed by my Otolaryngologist in Denver for extreme sensitivity to mold. However, for a while, I stopped taking the pills. I was diagnosed with RA in September of 2014. Inflammation levels were *extremely* high. I resumed taking the 300 mg capsules last year following your recommendation. Two weeks ago, I was retested and the blood test results were remarkable because all of the tests were negative in all RA categories and inflammation levels were normal. I believe that the Acetyl-Glutathione capsules and balm have helped in lowering the inflammation levels and pain. I highly recommend this product. -TL
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CitriSafe Glutathione Fact Sheet (PDF) |
Additional information
| Weight | 4 oz |
|---|---|
| Dimensions | 2.0 × 1.5 × 3.0 in |








